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Description

U-47700 is an opioid analgesic that acts as a selective agonist of the µ-opioid receptor with a Kd value of 5.3 nM compared to 910 nM for the κ-opioid receptor and has around 7.5 x the potency of morphine in animal models.

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U-47700 Powder is a synthetic opioid known for its potent analgesic effects. It is structurally related to fentanyl and is used in research and, in some cases, illicitly due to its powerful effects.

Chemical Overview:

  • Chemical Name: U-47700
  • Molecular Formula: C16H22N2O
  • CAS Number: 576-03-0
  • Appearance: White crystalline powder
  • Purity: 98%

U-47700 Powder is recognized for its white crystalline appearance and 98% purity, ensuring high-quality standards for research purposes.

Uses and Effects:

U-47700 is primarily used in research contexts:

  • Pain Relief: Known for its effectiveness in managing severe pain, similar to other opioids.
  • Research: Studied for its pharmacological effects and potential therapeutic applications.

Potential Side Effects:

Due to its potent opioid nature, U-47700 can cause a range of side effects:

  • Respiratory Depression: Risk of breathing difficulties or cessation.
  • Nausea and Vomiting: Common side effects associated with opioid use.
  • Drowsiness and Sedation: Can impair cognitive and motor functions.
  • Constipation: A frequent side effect of opioid use.
  • Addiction and Overdose Risk: High potential for dependency and overdose.

Dosage Information:

Dosage must be strictly controlled:

  • Pain Management: Typically requires precise dosing to avoid adverse effects.
  • Research Use: Doses vary based on experimental protocols and goals.

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